Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50216983 (CHEMBL392269 | UMB-96 | UMB96) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Maryland Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from cloned mu opioid receptor expressed in CHO cell membrane | Bioorg Med Chem Lett 17: 4829-31 (2007) Article DOI: 10.1016/j.bmcl.2007.06.050 BindingDB Entry DOI: 10.7270/Q2C8291Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Homo sapiens (Human)) | BDBM50216983 (CHEMBL392269 | UMB-96 | UMB96) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 89 | n/a | n/a | n/a | n/a |
University of Maryland Curated by ChEMBL | Assay Description Agonist activity at human mu opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assay | Bioorg Med Chem Lett 17: 4829-31 (2007) Article DOI: 10.1016/j.bmcl.2007.06.050 BindingDB Entry DOI: 10.7270/Q2C8291Q | |||||||||||
More data for this Ligand-Target Pair |