Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50008071 (5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents | Article PubMed | 6.92E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Firenze Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by liquid scintillation counter | J Med Chem 51: 3905-12 (2008) Article DOI: 10.1021/jm800145d BindingDB Entry DOI: 10.7270/Q2TX3GMC | |||||||||||
More data for this Ligand-Target Pair |