Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
NPC intracellular cholesterol transporter 1 (Homo sapiens (Human)) | BDBM50501737 (CHEMBL1091524) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Chaperone activity at FLAG/GFP-tagged NPC1 I1061T mutant (unknown origin) expressed in HEK293 cells assessed as increase in localization of protein m... | Bioorg Med Chem Lett 27: 2781-2787 (2017) Article DOI: 10.1016/j.bmcl.2017.04.062 BindingDB Entry DOI: 10.7270/Q2RX9G39 | |||||||||||
More data for this Ligand-Target Pair |