Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neprilysin (Mus musculus) | BDBM50027522 (2-(2-Carboxy-3-phenyl-propionylamino)-4-methyl-pen...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description 50% Inhibitory potency against enkephalinase from mouse striatum. | J Med Chem 26: 60-5 (1983) BindingDB Entry DOI: 10.7270/Q2Q81DP6 | |||||||||||
More data for this Ligand-Target Pair |