Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuraminidase (Influenza A virus) | BDBM50496023 (CHEMBL3120197) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
Christian-Albrechts University of Kiel Curated by ChEMBL | Assay Description Inhibition of neuraminidase in Influenza A virus A/HH/1580/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate a... | J Med Chem 57: 759-69 (2014) Article DOI: 10.1021/jm401492x BindingDB Entry DOI: 10.7270/Q21R6TG0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuraminidase (Influenza A virus) | BDBM50496023 (CHEMBL3120197) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.440 | n/a | n/a | n/a | n/a | n/a | n/a |
Christian-Albrechts University of Kiel Curated by ChEMBL | Assay Description Inhibition of neuraminidase in Influenza A virus A/Jena/5555/09(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate... | J Med Chem 57: 759-69 (2014) Article DOI: 10.1021/jm401492x BindingDB Entry DOI: 10.7270/Q21R6TG0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuraminidase (Influenza A virus) | BDBM50496023 (CHEMBL3120197) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.450 | n/a | n/a | n/a | n/a | n/a | n/a |
Christian-Albrechts University of Kiel Curated by ChEMBL | Assay Description Inhibition of neuraminidase in Influenza A virus A/Jena/5258/2009(H1N1) using Na-star as substrate preincubated for 10 to 30 mins followed by substra... | J Med Chem 57: 759-69 (2014) Article DOI: 10.1021/jm401492x BindingDB Entry DOI: 10.7270/Q21R6TG0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuraminidase (Influenza A virus) | BDBM50496023 (CHEMBL3120197) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Christian-Albrechts University of Kiel Curated by ChEMBL | Assay Description Inhibition of neuraminidase in Influenza A virus A/Berlin/10/04(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate... | J Med Chem 57: 759-69 (2014) Article DOI: 10.1021/jm401492x BindingDB Entry DOI: 10.7270/Q21R6TG0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuraminidase (Influenza A virus) | BDBM50496023 (CHEMBL3120197) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Christian-Albrechts University of Kiel Curated by ChEMBL | Assay Description Inhibition of neuraminidase in Influenza A virus A/Rheinland-Pfalz/3911/03(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed b... | J Med Chem 57: 759-69 (2014) Article DOI: 10.1021/jm401492x BindingDB Entry DOI: 10.7270/Q21R6TG0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuraminidase (Influenza A virus) | BDBM50496023 (CHEMBL3120197) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Christian-Albrechts University of Kiel Curated by ChEMBL | Assay Description Inhibition of neuraminidase in Influenza A virus A/Hong Kong/68(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate... | J Med Chem 57: 759-69 (2014) Article DOI: 10.1021/jm401492x BindingDB Entry DOI: 10.7270/Q21R6TG0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuraminidase (Influenza A virus) | BDBM50496023 (CHEMBL3120197) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Christian-Albrechts University of Kiel Curated by ChEMBL | Assay Description Inhibition of neuraminidase in Influenza A virus A/Sachsen/6/02(H3N2) using Na-star as substrate preincubated for 10 to 30 mins followed by substrate... | J Med Chem 57: 759-69 (2014) Article DOI: 10.1021/jm401492x BindingDB Entry DOI: 10.7270/Q21R6TG0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuraminidase (Influenza A virus) | BDBM50496023 (CHEMBL3120197) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Christian-Albrechts University of Kiel Curated by ChEMBL | Assay Description Inhibition of neuraminidase H274Y mutant in Oseltamivir-resistant Influenza A virus A/Berlin/55/08(H1N1) using Na-star as substrate preincubated for ... | J Med Chem 57: 759-69 (2014) Article DOI: 10.1021/jm401492x BindingDB Entry DOI: 10.7270/Q21R6TG0 | |||||||||||
More data for this Ligand-Target Pair |