Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuronal acetylcholine receptor subunit alpha-7 (Homo sapiens (Human)) | BDBM50025028 (CHEMBL3337866) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 813 | n/a | n/a | n/a | n/a | n/a | n/a |
The German University in Cairo Curated by ChEMBL | Assay Description Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assay | J Nat Prod 77: 2006-13 (2014) Article DOI: 10.1021/np500259j BindingDB Entry DOI: 10.7270/Q2H70HD8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuronal acetylcholine receptor subunit alpha-7 (Homo sapiens (Human)) | BDBM50025028 (CHEMBL3337866) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 820 | n/a | n/a | n/a | n/a | n/a | n/a |
The German University in Cairo Curated by ChEMBL | Assay Description Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assay | J Nat Prod 77: 2006-13 (2014) Article DOI: 10.1021/np500259j BindingDB Entry DOI: 10.7270/Q2H70HD8 | |||||||||||
More data for this Ligand-Target Pair |