Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50109185 (4-[3-(3-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of binding of [125I]-PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membrane | Bioorg Med Chem Lett 12: 379-82 (2002) BindingDB Entry DOI: 10.7270/Q2DJ5DZ8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50109185 (4-[3-(3-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of binding of [125I]-PYY to membranes of SK-N-MC cells expressing the human Y1 receptors | Bioorg Med Chem Lett 14: 5975-8 (2004) Article DOI: 10.1016/j.bmcl.2004.10.005 BindingDB Entry DOI: 10.7270/Q2765DTG | |||||||||||
More data for this Ligand-Target Pair |