Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Nischarin (RAT) | BDBM50473241 (CHEMBL288951) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article | 513 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to I1 imidazoline binding site in Rattus norvegicus (rat) PC12 cells | Citation and Details Article DOI: 10.1007/s00044-004-0023-9 BindingDB Entry DOI: 10.7270/Q2FJ2KNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nischarin (Homo sapiens (Human)) | BDBM50473241 (CHEMBL288951) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | 513 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Louis Pasteur Curated by ChEMBL | Assay Description Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranes | J Med Chem 44: 1588-93 (2001) Article DOI: 10.1021/jm001111b BindingDB Entry DOI: 10.7270/Q24M979D | |||||||||||
More data for this Ligand-Target Pair |