Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Norepinephrine transporter (RAT) | BDBM50029150 (3-(2-Piperidin-4-yl-ethyl)-1H-indole | CHEMBL27652...) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | PubMed | 513 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
McNeil Pharmaceutical Curated by PDSP Ki Database | J Pharmacol Exp Ther 247: 1032-8 (1988) BindingDB Entry DOI: 10.7270/Q2S75DV7 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Norepinephrine transporter (RAT) | BDBM50029150 (3-(2-Piperidin-4-yl-ethyl)-1H-indole | CHEMBL27652...) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 2.76E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
McGill University Curated by PDSP Ki Database | Eur J Pharmacol 349: 129-32 (1998) Article DOI: 10.1016/s0014-2999(98)00241-6 BindingDB Entry DOI: 10.7270/Q279436B | ||||||||||||
More data for this Ligand-Target Pair |