Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Nuclear receptor coactivator 2 [740-753]' and Ligand = 'BDBM205024'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Nuclear receptor coactivator 2 [740-753] ()	BDBM205024 (US9550781, 21 | n-(3-(3-(9h-purin-6-yl)pyridin-2-y...) Show SMILES Fc1ccc(NS(=O)(=O)C2CC2c2ccccc2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<500	n/a	n/a	n/a	n/a	n/a	n/a
Centaurus Biopharma Co., Ltd.; Chia Tai Tianqing Pharmaceutical Group Co., Ltd. US Patent					Assay Description In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...				US Patent US9550781 (2017) BindingDB Entry DOI: 10.7270/Q2X63PXK
					More data for this Ligand-Target Pair