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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Oxysterols receptor LXR-beta' and Ligand = 'BDBM27332'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Oxysterols receptor LXR-beta


(Homo sapiens (Human))		BDBM27332
PNG
(indole derivative, 38 | tert-butyl 2-{2-[(2-fluoro...)
Show SMILES CC(C)(C)OC(=O)n1c(cc2ccccc12)-c1ccc2CC(Cc2c1)NC(=O)c1ccccc1F
Show InChI InChI=1S/C29H27FN2O3/c1-29(2,3)35-28(34)32-25-11-7-4-8-19(25)17-26(32)20-13-12-18-15-22(16-21(18)14-20)31-27(33)23-9-5-6-10-24(23)30/h4-14,17,22H,15-16H2,1-3H3,(H,31,33)
PDB

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Similars
Article
PubMed
n/an/an/an/a 170n/an/an/an/a



Tanabe Research Laboratories USA



Assay Description
Polyhistidine-tagged human LXR ligand-binding domain was mixed with the test compound, biotin-SRC1 peptide, streptavidin-allophycocyanin, and europiu...

Bioorg Med Chem Lett 17: 3473-9 (2007)


Article DOI: 10.1016/j.bmcl.2007.03.076
BindingDB Entry DOI: 10.7270/Q2HD7T00
More data for this
Ligand-Target Pair