BindingDB PrimarySearch

Found 1 hit Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 12' and Ligand = 'BDBM50500441'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
P2Y purinoceptor 12 (Homo sapiens (Human))	BDBM50500441 (CHEMBL3746502) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	9.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
GLSynthesis, Inc. Curated by ChEMBL					Assay Description Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...				Eur J Med Chem 107: 204-18 (2016) Article DOI: 10.1016/j.ejmech.2015.10.055 BindingDB Entry DOI: 10.7270/Q2PN98NM
GLSynthesis, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair