BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50248411'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human))	BDBM50248411 (5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pheny...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Bristol-Myers Squibb Research and Development Curated by ChEMBL					Assay Description Binding affinity to PPARalpha (unknown origin) by fluorescence polarization assay				Bioorg Med Chem Lett 19: 1451-6 (2009) Article DOI: 10.1016/j.bmcl.2009.01.030 BindingDB Entry DOI: 10.7270/Q2MC8ZW8
					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human))	BDBM50248411 (5-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pheny...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	>1.50E+4	n/a	n/a	n/a	n/a
Bristol-Myers Squibb Research and Development Curated by ChEMBL					Assay Description Agonist activity at human PPARalpha ligand binding domain expressed in HEK293 cells by Gal4 transactivation assay				Bioorg Med Chem Lett 19: 1451-6 (2009) Article DOI: 10.1016/j.bmcl.2009.01.030 BindingDB Entry DOI: 10.7270/Q2MC8ZW8
					More data for this Ligand-Target Pair