Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM50508142 (CHEMBL4452945) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 515 | n/a | n/a | n/a | n/a | n/a | n/a |
Inception Sciences Curated by ChEMBL | Assay Description Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba... | Bioorg Med Chem Lett 29: 503-508 (2019) Article DOI: 10.1016/j.bmcl.2018.12.045 BindingDB Entry DOI: 10.7270/Q2XK8JVQ | |||||||||||
More data for this Ligand-Target Pair |