Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM50309074 (2-(4-fluorophenyl)-11-phenyl-4,9-dioxa-3,10-diazat...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a |
Zydus Research Centre Curated by ChEMBL | Assay Description Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos... | Bioorg Med Chem Lett 20: 1156-61 (2010) Article DOI: 10.1016/j.bmcl.2009.12.022 BindingDB Entry DOI: 10.7270/Q20865FJ | |||||||||||
More data for this Ligand-Target Pair |