Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM50317118 ((S)-2-(methoxycarbonyl(1-(3-((2-p-tolyloxazol-4-yl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.07E+4 | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb R&D Curated by ChEMBL | Assay Description Agonist activity against human Gal4-fussed PPARgamma in HEK293 cells by luciferase reporter gene assay | Bioorg Med Chem Lett 20: 2933-7 (2010) Article DOI: 10.1016/j.bmcl.2010.03.019 BindingDB Entry DOI: 10.7270/Q2K35TS2 | |||||||||||
More data for this Ligand-Target Pair |