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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147]' and Ligand = 'BDBM222683'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Peroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147]


(Saccharomyces bayanus (Yeast)-Homo sapiens (Human))		BDBM222683
PNG
(US9315493, 15)
Show SMILES CCCCc1nc(C)n(-c2cc(C)ccn2)c(=O)c1Cc1ccc(nc1)-c1ccccc1-c1noc(=O)[nH]1
Show InChI InChI=1S/C29H28N6O3/c1-4-5-10-25-23(28(36)35(19(3)32-25)26-15-18(2)13-14-30-26)16-20-11-12-24(31-17-20)21-8-6-7-9-22(21)27-33-29(37)38-34-27/h6-9,11-15,17H,4-5,10,16H2,1-3H3,(H,33,34,37)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 3.61E+3n/an/an/an/a



KOWA COMPANY, LTD.

US Patent


Assay Description
As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...

US Patent US9315493 (2016)


BindingDB Entry DOI: 10.7270/Q27M06SS
More data for this
Ligand-Target Pair