Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Phosphatidylinositol 4-kinase beta (Homo sapiens (Human)) | BDBM50005005 (CHEMBL2397317) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Pharma Curated by ChEMBL | Assay Description Inhibition of recombinant human full length GST-tagged PI4K3beta expressed in baculovirus expression system using PI lipid kinase substrate after 60 ... | J Med Chem 61: 6705-6723 (2018) Article DOI: 10.1021/acs.jmedchem.8b00521 BindingDB Entry DOI: 10.7270/Q2FF3W01 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phosphatidylinositol 4-kinase beta (Homo sapiens (Human)) | BDBM50005005 (CHEMBL2397317) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
BioFocus Curated by ChEMBL | Assay Description Inhibition of PI4K3beta (unknown origin) | ACS Med Chem Lett 4: 585-9 (2013) Article DOI: 10.1021/ml400095m BindingDB Entry DOI: 10.7270/Q2N58Q8J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phosphatidylinositol 4-kinase beta (Homo sapiens (Human)) | BDBM50005005 (CHEMBL2397317) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 137 | n/a | n/a | n/a | n/a | n/a | n/a |
Boehringer Ingelheim (Canada) Ltd. Curated by ChEMBL | Assay Description Inhibition of PI4K3beta (unknown origin) | Bioorg Med Chem Lett 23: 3841-7 (2013) Article DOI: 10.1016/j.bmcl.2013.04.077 BindingDB Entry DOI: 10.7270/Q2BG2QCX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phosphatidylinositol 4-kinase beta (Homo sapiens (Human)) | BDBM50005005 (CHEMBL2397317) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Pharma Curated by ChEMBL | Assay Description Inhibition of PI4K3beta in human PBMC assessed as reduction in mitomycin-C treated human RPMI1788 cells-stimulated lymphocyte proliferation by measur... | J Med Chem 61: 6705-6723 (2018) Article DOI: 10.1021/acs.jmedchem.8b00521 BindingDB Entry DOI: 10.7270/Q2FF3W01 | |||||||||||
More data for this Ligand-Target Pair |