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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50018322'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50018322
PNG
(4,4''-Dimethoxy-[1,1';2',1'']terphenyl-4'-carboxyl...)
Show SMILES COc1ccc(cc1)-c1ccc(cc1-c1ccc(OC)cc1)C(=O)NCCCCc1cccnc1
Show InChI InChI=1S/C30H30N2O3/c1-34-26-13-8-23(9-14-26)28-17-12-25(20-29(28)24-10-15-27(35-2)16-11-24)30(33)32-19-4-3-6-22-7-5-18-31-21-22/h5,7-18,20-21H,3-4,6,19H2,1-2H3,(H,32,33)
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Roche Research Center

Curated by ChEMBL


Assay Description
Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.

J Med Chem 32: 1814-20 (1989)


BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ
More data for this
Ligand-Target Pair