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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50018333'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50018333
PNG
(2,3',4'-Trimethoxy-biphenyl-4-carboxylic acid (4-p...)
Show SMILES COc1ccc(cc1OC)-c1ccc(cc1OC)C(=O)NCCCCc1cccnc1
Show InChI InChI=1S/C25H28N2O4/c1-29-22-12-10-19(15-24(22)31-3)21-11-9-20(16-23(21)30-2)25(28)27-14-5-4-7-18-8-6-13-26-17-18/h6,8-13,15-17H,4-5,7,14H2,1-3H3,(H,27,28)
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Roche Research Center

Curated by ChEMBL


Assay Description
Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.

J Med Chem 32: 1814-20 (1989)


BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ
More data for this
Ligand-Target Pair