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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50018348'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50018348
PNG
(5,5-Bis-(3,4-dimethoxy-phenyl)-penta-2,4-dienoic a...)
Show SMILES [#6]-[#8]-c1ccc(cc1-[#8]-[#6])-[#6](=[#6]/[#6]=[#6]/[#6](=O)-[#7]-[#6]-[#6]-[#6]-[#6]-c1cccnc1)\c1ccc(-[#8]-[#6])c(-[#8]-[#6])c1
Show InChI InChI=1S/C30H34N2O5/c1-34-26-15-13-23(19-28(26)36-3)25(24-14-16-27(35-2)29(20-24)37-4)11-7-12-30(33)32-18-6-5-9-22-10-8-17-31-21-22/h7-8,10-17,19-21H,5-6,9,18H2,1-4H3,(H,32,33)/b12-7+
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PubMed
n/an/a 55n/an/an/an/an/an/a



Roche Research Center

Curated by ChEMBL


Assay Description
Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand

J Med Chem 32: 1820-35 (1989)


BindingDB Entry DOI: 10.7270/Q2NZ86MR
More data for this
Ligand-Target Pair