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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50282039'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50282039
PNG
(1-{2-[5-(3,4-Dimethoxy-phenyl)-tetrahydro-furan-2-...)
Show SMILES COc1ccc(cc1OC)C1CCC(COCCn2c(C)nc3cnccc23)O1
Show InChI InChI=1S/C22H27N3O4/c1-15-24-18-13-23-9-8-19(18)25(15)10-11-28-14-17-5-7-20(29-17)16-4-6-21(26-2)22(12-16)27-3/h4,6,8-9,12-13,17,20H,5,7,10-11,14H2,1-3H3
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TBA

Curated by ChEMBL


Assay Description
Inhibition of [3H]PAF receptor binding to washed human platelet membranes determined in vitro

Bioorg Med Chem Lett 3: 1499-1504 (1993)


Article DOI: 10.1016/S0960-894X(00)80006-2
BindingDB Entry DOI: 10.7270/Q2CC115V
More data for this
Ligand-Target Pair