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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50286658'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50286658
PNG
(5-lipoxygenase inhibitor | CHEMBL155760)
Show SMILES CCCOc1cc(cc(N(CC)C(=O)N(O)CCC)c1OCCC)[C@H]1CC[C@@H](O1)c1cc(OC)c(OC)c(OC)c1
Show InChI InChI=1S/C31H46N2O8/c1-8-14-33(35)31(34)32(11-4)23-17-21(20-28(39-15-9-2)29(23)40-16-10-3)24-12-13-25(41-24)22-18-26(36-5)30(38-7)27(19-22)37-6/h17-20,24-25,35H,8-16H2,1-7H3/t24-,25-/m1/s1
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Similars
Article
n/an/a 56n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.

Bioorg Med Chem Lett 5: 643-648 (1995)


Article DOI: 10.1016/0960-894X(95)00088-B
BindingDB Entry DOI: 10.7270/Q23778QB
More data for this
Ligand-Target Pair