Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-derived growth factor receptor alpha (Homo sapiens (Human)) | BDBM4810 ((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Microbial Chemistry (BIKAKEN) Curated by ChEMBL | Assay Description Inhibition of PDGFR-alpha (unknown origin) after 20 mins by scintillation counting | J Nat Prod 76: 715-9 (2013) Article DOI: 10.1021/np300535c BindingDB Entry DOI: 10.7270/Q2JQ12BH | |||||||||||
More data for this Ligand-Target Pair |