Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Polycystin-1 (Homo sapiens (Human)) | BDBM86435 (B8-DL-B8 | B8-DL-B8 (low PS)) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 10.8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pittsburgh Curated by PDSP Ki Database | Mol Pharmacol 64: 1342-8 (2003) Article DOI: 10.1124/mol.64.6.1342 BindingDB Entry DOI: 10.7270/Q270800T | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polycystin-1 (Homo sapiens (Human)) | BDBM86435 (B8-DL-B8 | B8-DL-B8 (low PS)) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 26.1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Pittsburgh Curated by PDSP Ki Database | Mol Pharmacol 64: 1342-8 (2003) Article DOI: 10.1124/mol.64.6.1342 BindingDB Entry DOI: 10.7270/Q270800T | ||||||||||||
More data for this Ligand-Target Pair |