Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human)) | BDBM50371942 (CHEMBL272101) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
The Walter and Eliza Hall Institute of Medical Research Curated by ChEMBL | Assay Description Inhibition in Kv1.3 expressed in human Jurkat cells by patch clamp method | Bioorg Med Chem Lett 18: 2055-61 (2008) Article DOI: 10.1016/j.bmcl.2008.01.099 BindingDB Entry DOI: 10.7270/Q2ZG6T27 | |||||||||||
More data for this Ligand-Target Pair |