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Found 1 hit Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 5' and Ligand = 'BDBM50198247'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Potassium voltage-gated channel subfamily A member 5


(Homo sapiens (Human))		BDBM50198247
PNG
(2-(3,4-dimethylphenyl)-3-(4-methoxyphenethyl)-2-me...)
Show SMILES COc1ccc(CCN2C(=O)CSC2(C)c2ccc(C)c(C)c2)cc1
Show InChI InChI=1S/C21H25NO2S/c1-15-5-8-18(13-16(15)2)21(3)22(20(23)14-25-21)12-11-17-6-9-19(24-4)10-7-17/h5-10,13H,11-12,14H2,1-4H3
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Similars
Article
PubMed
n/an/a 69n/an/an/an/an/an/a



Procter and Gamble Pharmaceuticals

Curated by ChEMBL


Assay Description
Inhibition of Kv1.5 mediated ultra-rapid delayed rectifier current Ikur in human atrial cells

Bioorg Med Chem Lett 17: 282-4 (2006)


Article DOI: 10.1016/j.bmcl.2006.07.007
BindingDB Entry DOI: 10.7270/Q2S18256
More data for this
Ligand-Target Pair