Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50199060 (4-(3-fluorophenyl)-6-methoxy-1-(4-methyl-1H-imidaz...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Antagonist activity at human Kv1.5 channel expressed in CHO cell membrane by HT clamp assay | J Med Chem 49: 6954-7 (2006) Article DOI: 10.1021/jm060927v BindingDB Entry DOI: 10.7270/Q2ST7PG7 | |||||||||||
More data for this Ligand-Target Pair |