Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50385911 (CHEMBL531475 | TCMDC-133351) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cape Town Curated by ChEMBL | Assay Description Inhibition of human ERG expressed in CHO cells by IonWorks assay | J Med Chem 55: 3479-87 (2012) Article DOI: 10.1021/jm3001373 BindingDB Entry DOI: 10.7270/Q2V125T9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50385911 (CHEMBL531475 | TCMDC-133351) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cape Town Curated by ChEMBL | Assay Description Inhibition of human ERG channel expressed in Chinese hamster lung cells after 6 to 7 mins by patch clamp assay | J Med Chem 56: 7750-4 (2013) Article DOI: 10.1021/jm400279y BindingDB Entry DOI: 10.7270/Q23R0WS6 | |||||||||||
More data for this Ligand-Target Pair |