Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50509618 (CHEMBL4463663) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.78E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Korea Research Institute of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of human ERG expressed in human HEK293 cells by patch clamp assay | ACS Med Chem Lett 11: 166-171 (2020) Article DOI: 10.1021/acsmedchemlett.9b00550 BindingDB Entry DOI: 10.7270/Q2RF5Z9F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50509618 (CHEMBL4463663) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.09E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Korea Research Institute of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of human ERG by competitive fluorescence polarization assay | ACS Med Chem Lett 11: 166-171 (2020) Article DOI: 10.1021/acsmedchemlett.9b00550 BindingDB Entry DOI: 10.7270/Q2RF5Z9F | |||||||||||
More data for this Ligand-Target Pair |