Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50534415 (CHEMBL4464764) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 9.93E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Modena and Reggio Emilia Curated by ChEMBL | Assay Description Inhibition of human ERG in membranes incubated for 2 hrs by fluorescence polarization assay | J Med Chem 59: 7598-616 (2016) Article DOI: 10.1021/acs.jmedchem.6b00698 BindingDB Entry DOI: 10.7270/Q25D8WBK | |||||||||||
More data for this Ligand-Target Pair |