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Found 1 hit Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily KQT member 1' and Ligand = 'BDBM50106171'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Potassium voltage-gated channel subfamily KQT member 1


(Cavia porcellus)		BDBM50106171
PNG
(CHEMBL122637 | Diethyl-{2-[4-(1,1,3,3-tetramethyl-...)
Show SMILES CCN(CC)CCOc1ccc(cc1)C(C)(C)CC(C)(C)C
Show InChI InChI=1S/C20H35NO/c1-8-21(9-2)14-15-22-18-12-10-17(11-13-18)20(6,7)16-19(3,4)5/h10-13H,8-9,14-16H2,1-7H3
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars
PubMed
n/an/a 5.00E+3n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytes

J Med Chem 44: 3764-7 (2001)


BindingDB Entry DOI: 10.7270/Q2G1604C
More data for this
Ligand-Target Pair