Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily KQT member 4 (Homo sapiens (Human)) | BDBM50526876 (CHEMBL4457044) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a |
University Federico II of Naples Curated by ChEMBL | Assay Description Activation of human Kv7.4 expressed in CHO cells assessed as increase in channel current amplitude by whole cell patch clamp electrophysiology assay | J Med Chem 63: 163-185 (2020) Article DOI: 10.1021/acs.jmedchem.9b00796 BindingDB Entry DOI: 10.7270/Q2KW5KG2 | |||||||||||
More data for this Ligand-Target Pair |