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Compile Data Set for Download or QSAR

Found 2 hits Enz. Inhib. hit(s) with Target = 'Probable G-protein coupled receptor 142' and Ligand = 'BDBM50558203'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558203
PNG
(CHEMBL4751866)
Show SMILES COc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>2.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558203
PNG
(CHEMBL4751866)
Show SMILES COc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>2.00E+4n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair