BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Prokineticin receptor 1' and Ligand = 'BDBM347528'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Prokineticin receptor 1


(Homo sapiens (Human))
BDBM347528
PNG
(N,N-Dimethyl-4-{[3-(2-methylphenyl)piperidin-1-yl]...)
Show SMILES CN(C)c1cc(ccn1)C(=O)N1CCCC(C1)c1ccccc1C
Show InChI InChI=1S/C20H25N3O/c1-15-7-4-5-9-18(15)17-8-6-12-23(14-17)20(24)16-10-11-21-19(13-16)22(2)3/h4-5,7,9-11,13,17H,6,8,12,14H2,1-3H3
MMDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 190n/an/an/an/an/an/a



Takeda Pharmaceutical Company Limited

US Patent


Assay Description
Prokineticin receptor 1 (PKR1) antagonists may be functionally assessed by measurement of change in intracellular calcium levels induced by Gq mediat...


US Patent US9790201 (2017)


BindingDB Entry DOI: 10.7270/Q2377BVZ
More data for this
Ligand-Target Pair