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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Prokineticin receptor 1' and Ligand = 'BDBM347579'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Prokineticin receptor 1


(Homo sapiens (Human))		BDBM347579
PNG
(4-{[3-(4-Chloro-2-ethoxyphenyl)piperidin-1-yl]carb...)
Show SMILES CCOc1cc(Cl)ccc1C1CCCN(C1)C(=O)c1ccnc(NC)c1
Show InChI InChI=1S/C20H24ClN3O2/c1-3-26-18-12-16(21)6-7-17(18)15-5-4-10-24(13-15)20(25)14-8-9-23-19(11-14)22-2/h6-9,11-12,15H,3-5,10,13H2,1-2H3,(H,22,23)
MMDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
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PC cid
PC sid
UniChem
US Patent
n/an/a 70n/an/an/an/an/an/a



Takeda Pharmaceutical Company Limited

US Patent


Assay Description
Prokineticin receptor 1 (PKR1) antagonists may be functionally assessed by measurement of change in intracellular calcium levels induced by Gq mediat...

US Patent US9790201 (2017)


BindingDB Entry DOI: 10.7270/Q2377BVZ
More data for this
Ligand-Target Pair