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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Prokineticin receptor 1' and Ligand = 'BDBM347580'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Prokineticin receptor 1


(Homo sapiens (Human))		BDBM347580
PNG
(4-({3-[2-(Difluoromethoxy)phenyl]piperidin-1-yl}ca...)
Show SMILES CN(C)c1cc(ccn1)C(=O)N1CCCC(C1)c1ccccc1OC(F)F
Show InChI InChI=1S/C20H23F2N3O2/c1-24(2)18-12-14(9-10-23-18)19(26)25-11-5-6-15(13-25)16-7-3-4-8-17(16)27-20(21)22/h3-4,7-10,12,15,20H,5-6,11,13H2,1-2H3
MMDB

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US Patent
n/an/a 700n/an/an/an/an/an/a



Takeda Pharmaceutical Company Limited

US Patent


Assay Description
Prokineticin receptor 1 (PKR1) antagonists may be functionally assessed by measurement of change in intracellular calcium levels induced by Gq mediat...

US Patent US9790201 (2017)


BindingDB Entry DOI: 10.7270/Q2377BVZ
More data for this
Ligand-Target Pair