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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Prokineticin receptor 1' and Ligand = 'BDBM347594'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Prokineticin receptor 1


(Homo sapiens (Human))		BDBM347594
PNG
(5-{[3-(4-Methoxy-2-methylphenyl)piperidin-1-yl]car...)
Show SMILES CNc1cc(cnn1)C(=O)N1CCCC(C1)c1ccc(OC)cc1C
Show InChI InChI=1S/C19H24N4O2/c1-13-9-16(25-3)6-7-17(13)14-5-4-8-23(12-14)19(24)15-10-18(20-2)22-21-11-15/h6-7,9-11,14H,4-5,8,12H2,1-3H3,(H,20,22)
MMDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
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PC cid
PC sid
UniChem
US Patent
n/an/a 130n/an/an/an/an/an/a



Takeda Pharmaceutical Company Limited

US Patent


Assay Description
Prokineticin receptor 1 (PKR1) antagonists may be functionally assessed by measurement of change in intracellular calcium levels induced by Gq mediat...

US Patent US9790201 (2017)


BindingDB Entry DOI: 10.7270/Q2377BVZ
More data for this
Ligand-Target Pair