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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Prokineticin receptor 2' and Ligand = 'BDBM463306'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Prokineticin receptor 2


(Homo sapiens (Human))		BDBM463306
PNG
((-)-(2R)-1-(4-Fluoro-3- methoxybenzyl)-N-(9-chloro...)
Show SMILES COc1cc(CN2CCOC(C2)C(=O)N(CC(C)C)Cc2cc(Cl)c3OCCCOc3c2)ccc1F
Show InChI InChI=1S/C27H34ClFN2O5/c1-18(2)14-31(16-20-11-21(28)26-24(13-20)34-8-4-9-36-26)27(32)25-17-30(7-10-35-25)15-19-5-6-22(29)23(12-19)33-3/h5-6,11-13,18,25H,4,7-10,14-17H2,1-3H3
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US Patent
 1.90n/an/an/an/an/an/an/an/a



THE REGENTS OF THE UNIVERSITY OF CALIFORNIA

US Patent


Assay Description
An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...

US Patent US10780095 (2020)


BindingDB Entry DOI: 10.7270/Q22F7RH6
More data for this
Ligand-Target Pair