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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-5' and Ligand = 'BDBM50185650'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Proteasome subunit beta type-5


(Saccharomyces cerevisiae)		BDBM50185650
PNG
(CHEMBL209568 | Pam-YET)
Show SMILES CCCCCCCCCCCCCCCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H]([C@@H](C)O)C(O)=O
Show InChI InChI=1S/C34H55N3O9/c1-3-4-5-6-7-8-9-10-11-12-13-14-15-16-29(40)35-28(23-25-17-19-26(39)20-18-25)33(44)36-27(21-22-30(41)42)32(43)37-31(24(2)38)34(45)46/h17-20,24,27-28,31,38-39H,3-16,21-23H2,1-2H3,(H,35,40)(H,36,44)(H,37,43)(H,41,42)(H,45,46)/t24-,27+,28+,31+/m1/s1
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Similars
Article
PubMed
 2.00E+4n/an/an/an/an/an/an/an/a



CNRS-Université Paris VI

Curated by ChEMBL


Assay Description
Inhibition of chymotrypsin like activity of yeast 20S proteasome

Bioorg Med Chem Lett 16: 3277-81 (2006)


Article DOI: 10.1016/j.bmcl.2006.03.033
BindingDB Entry DOI: 10.7270/Q280527Z
More data for this
Ligand-Target Pair