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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha/beta/gamma type' and Ligand = 'BDBM50229917'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Protein kinase C alpha/beta/gamma type


(Rattus norvegicus (Rat)-Rattus norvegicus (rat))		BDBM50229917
PNG
(CHEMBL100289)
Show SMILES [H][C@](N)(CCCCN)C(=O)NCC1CCCCN1C(=O)CCCCCCCCCCCCCCC
Show InChI InChI=1S/C28H56N4O2/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-21-27(33)32-23-18-16-19-25(32)24-31-28(34)26(30)20-15-17-22-29/h25-26H,2-24,29-30H2,1H3,(H,31,34)/t25?,26-/m0/s1
PDB

UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem
PubMed
n/an/a 4.50E+4n/an/an/an/an/an/a



Nova Pharmaceutical Corporation

Curated by ChEMBL


Assay Description
In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...

J Med Chem 34: 2928-31 (1991)


BindingDB Entry DOI: 10.7270/Q2KH0NZG
More data for this
Ligand-Target Pair