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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Protein kinase C beta type' and Ligand = 'BDBM2648'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Protein kinase C beta type


(Rattus norvegicus (rat))
BDBM2648
PNG
((Phenylindolyl)maleimide deriv. 70 | 3-(1-methyl-1...)
Show SMILES Cn1cc(C2=C(C(=O)NC2=O)c2cccc(c2)[N+]([O-])=O)c2ccccc12 |t:4|
Show InChI InChI=1S/C19H13N3O4/c1-21-10-14(13-7-2-3-8-15(13)21)17-16(18(23)20-19(17)24)11-5-4-6-12(9-11)22(25)26/h2-10H,1H3,(H,20,23,24)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Patents


Similars

Article
PubMed
n/an/a 1.90E+3n/an/an/an/an/an/a



Roche Products Limited



Assay Description
The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...


J Med Chem 35: 177-84 (1992)


Article DOI: 10.1021/jm00079a024
BindingDB Entry DOI: 10.7270/Q2K64G8V
More data for this
Ligand-Target Pair