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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Protein kinase C beta type' and Ligand = 'BDBM2653'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Protein kinase C beta type


(Rattus norvegicus (rat))		BDBM2653
PNG
((Phenylindolyl)maleimide deriv. 75 | 3-(1-methyl-1...)
Show SMILES Cn1cc(C2=C(C(=O)NC2=O)c2ccccc2C(F)(F)F)c2ccccc12 |t:4|
Show InChI InChI=1S/C20H13F3N2O2/c1-25-10-13(11-6-3-5-9-15(11)25)17-16(18(26)24-19(17)27)12-7-2-4-8-14(12)20(21,22)23/h2-10H,1H3,(H,24,26,27)
PDB

UniProtKB/SwissProt

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PC cid
PC sid
UniChem

Patents

Similars
Article
PubMed
n/an/a 950n/an/an/an/an/an/a



Roche Products Limited



Assay Description
The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...

J Med Chem 35: 177-84 (1992)


Article DOI: 10.1021/jm00079a024
BindingDB Entry DOI: 10.7270/Q2K64G8V
More data for this
Ligand-Target Pair