Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Protein kinase C beta type' and Ligand = 'BDBM2654'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Protein kinase C beta type (Rattus norvegicus (rat))	BDBM2654 ((Phenylindolyl)maleimide deriv. 76 | 3-(2,3-dimeth...) Show SMILES Cc1cccc(C2=C(C(=O)NC2=O)c2cn(C)c3ccccc23)c1C |t:6| Show InChI InChI=1S/C21H18N2O2/c1-12-7-6-9-14(13(12)2)18-19(21(25)22-20(18)24)16-11-23(3)17-10-5-4-8-15(16)17/h4-11H,1-3H3,(H,22,24,25)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	2.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
Roche Products Limited					Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...				J Med Chem 35: 177-84 (1992) Article DOI: 10.1021/jm00079a024 BindingDB Entry DOI: 10.7270/Q2K64G8V
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