BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Protein kinase C epsilon type' and Ligand = 'BDBM3240'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Protein kinase C epsilon type (Homo sapiens (Human))	BDBM3240 ((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article	n/a	n/a	3.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of Human Protein kinase C epsilon				Bioorg Med Chem Lett 5: 1839-1842 (1995) Article DOI: 10.1016/0960-894X(95)00303-B BindingDB Entry DOI: 10.7270/Q2QN66R9
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C epsilon type (Homo sapiens (Human))	BDBM3240 ((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
Sphinx Laboratories					Assay Description PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.				J Med Chem 45: 2624-43 (2002) Article DOI: 10.1021/jm020018f BindingDB Entry DOI: 10.7270/Q2BG2M50
Sphinx Laboratories					More data for this Ligand-Target Pair