Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein mono-ADP-ribosyltransferase PARP6 (Homo sapiens (Human)) | BDBM50434127 (CHEMBL2381633) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nanyang Technological University Curated by ChEMBL | Assay Description Inhibition of PARP6 (unknown origin) | J Med Chem 56: 4497-508 (2013) Article DOI: 10.1021/jm400211f BindingDB Entry DOI: 10.7270/Q23R0V82 | |||||||||||
More data for this Ligand-Target Pair |