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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Protein-tyrosine kinase 2-beta' and Ligand = 'BDBM286384'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Protein-tyrosine kinase 2-beta


(Homo sapiens (Human))		BDBM286384
PNG
(5-{[(2S,5R)-2,5-dimethyl-4-(tetrahydro-2H-pyran-4-...)
Show SMILES COCc1ncc(F)c(Nc2n[nH]c3c2CN(C(=O)C2C[C@@H](C)N(CC4CCOCC4)C[C@@H]2C)C3(C)C)n1 |r|
Show InChI InChI=1S/C27H40FN7O3/c1-16-12-34(13-18-6-8-38-9-7-18)17(2)10-19(16)26(36)35-14-20-23(27(35,3)4)32-33-24(20)31-25-21(28)11-29-22(30-25)15-37-5/h11,16-19H,6-10,12-15H2,1-5H3,(H2,29,30,31,32,33)/t16-,17+,19?/m0/s1
PDB

UniProtKB/SwissProt

antibodypedia
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PC cid
PC sid
UniChem
US Patent
<10n/an/an/an/an/an/a7.4n/a



PFIZER INC.

US Patent


Assay Description
Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...

US Patent US9518060 (2016)


BindingDB Entry DOI: 10.7270/Q2ZK5JPN
More data for this
Ligand-Target Pair