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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'RCG37580' and Ligand = 'BDBM16'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
RCG37580


(Rattus norvegicus)
BDBM16
PNG
(Zn2+ | zinc(2+) ion)
Show InChI InChI=1S/Zn/q+2
KEGG

UniProtKB/TrEMBL

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MCE
KEGG
MMDB
PC cid
PC sid
PDB
UniChem
Article
PubMed
n/an/an/an/a 4.04E+3n/an/an/an/a



Novartis Institutes for BioMedical Research

Curated by ChEMBL


Assay Description
Agonist activity at rat GPR39 expressed in HEK293 cells by IP1 assay


ACS Med Chem Lett 5: 1114-8 (2014)


Article DOI: 10.1021/ml500240d
BindingDB Entry DOI: 10.7270/Q2MC91MW
More data for this
Ligand-Target Pair