Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50122348 ((2E,4E)-6-[1-(3,5-Di-tert-butyl-phenyl)-cyclopropy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Transcriptional activation assay in CV-1 cells expressing human retinoid X receptor RXR alpha | Bioorg Med Chem Lett 13: 261-4 (2002) BindingDB Entry DOI: 10.7270/Q29P310V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50122348 ((2E,4E)-6-[1-(3,5-Di-tert-butyl-phenyl)-cyclopropy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | n/a | n/a | 733 | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Transcriptional activation in CV-1 cells expresing human Retinoic acid receptor RAR alpha | Bioorg Med Chem Lett 13: 261-4 (2002) BindingDB Entry DOI: 10.7270/Q29P310V | |||||||||||
More data for this Ligand-Target Pair |