Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Retinoic acid receptor gamma (Mus musculus) | BDBM50526314 (CHEMBL4459692 | US10752616, Code No. BHBA-001) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 13 | n/a | n/a | n/a | n/a |
King's College Curated by ChEMBL | Assay Description Transactivation of GAL4-fused mouse RARgamma-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assay | Bioorg Med Chem Lett 29: 995-1000 (2019) Article DOI: 10.1016/j.bmcl.2019.02.011 BindingDB Entry DOI: 10.7270/Q25142NC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoic acid receptor gamma (Homo sapiens (Human)) | BDBM50526314 (CHEMBL4459692 | US10752616, Code No. BHBA-001) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 11 | n/a | n/a | n/a | n/a |
King''s College London US Patent | Assay Description Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e... | US Patent US10752616 (2020) BindingDB Entry DOI: 10.7270/Q2B85C6M | |||||||||||
More data for this Ligand-Target Pair |